Design, Synthesis, and Evaluation of 2-Methyl- and 2-Amino-N-aryl-4,5-dihydrothiazolo[4,5-h]quinazolin-8-amines as Ring-Constrained 2-Anilino-4-(thiazol-5-yl)pyrimidine Cyclin-Dependent Kinase Inhibitors-Reference-Cited by-同舟云学术

Design, Synthesis, and Evaluation of 2-Methyl- and 2-Amino-N-aryl-4,5-dihydrothiazolo[4,5-h]quinazolin-8-amines as Ring-Constrained 2-Anilino-4-(thiazol-5-yl)pyrimidine Cyclin-Dependent Kinase Inhibitors

Published:2010-02-10 Issue:5 Volume:53 Page:2136-2145
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

McIntyre Neil A.¹,McInnes Campbell²,Griffiths Gary²,Barnett Anna L.²,Kontopidis George²,Slawin Alexandra M. Z.¹,Jackson Wayne²,Thomas Mark²,Zheleva Daniella I.²,Wang Shudong²,Blake David G.²,Westwood Nicholas J.¹,Fischer Peter M.²

Affiliation:

1. School of Chemistry and Biomedical Sciences Research Complex, University of St. Andrews, North Haugh, St. Andrews, Fife KY16 9ST, U.K.

2. Cyclacel Limited, 1 James Lindsay Place, Dundee DD1 5JJ, U.K

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm901660c

Reference43 articles.

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