Synthesis of a 3-(α-Styryl)benzo[b]-thiophene Library via Bromocyclization of Alkynes and Palladium-Catalyzed Tosylhydrazones Cross-Couplings: Evaluation as Antitubulin Agents-Reference-Cited by-同舟云学术

Synthesis of a 3-(α-Styryl)benzo[b]-thiophene Library via Bromocyclization of Alkynes and Palladium-Catalyzed Tosylhydrazones Cross-Couplings: Evaluation as Antitubulin Agents

Published:2014-09-25 Issue:12 Volume:16 Page:702-710
ISSN:2156-8952
Container-title:ACS Combinatorial Science
language:en
Short-container-title:ACS Comb. Sci.

Author:

Tréguier Bret¹,Lawson Marie¹,Bernadat Guillaume¹,Bignon Jérôme²,Dubois Joëlle²,Brion Jean-Daniel¹,Alami Mouad¹,Hamze Abdallah¹

Affiliation:

1. Univ Paris Sud, CNRS, BioCIS−UMR 8076, Laboratoire de Chimie Thérapeutique, Equipe Labellisée Ligue Contre le Cancer, LabEx LERMIT, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry, F-92296, France

2. Institut de Chimie des Substances Naturelles, UPR 2301, CNRS, avenue de la Terrasse, F-91198 Gif sur Yvette, France

Funder

Centre National de la Recherche Scientifique

Publisher

American Chemical Society (ACS)

Subject

General Chemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/co500115b

Reference52 articles.

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3. Microtubules as a target for anticancer drugs

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5. The binding conformation of Taxol in -tubulin: A model based on electron crystallographic density

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