Design, Synthesis, and Pharmacological Characterization of Novel Endomorphin-1 Analogues as Extremely Potent μ-Opioid Agonists-Reference-Cited by-同舟云学术

Design, Synthesis, and Pharmacological Characterization of Novel Endomorphin-1 Analogues as Extremely Potent μ-Opioid Agonists

Published:2013-03-28 Issue:7 Volume:56 Page:3102-3114
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Liu Xin¹,Wang Yuan¹,Xing Yanhong¹,Yu Jing¹,Ji Hong¹,Kai Ming¹,Wang Zilong¹,Wang Dan¹,Zhang Yixin¹,Zhao Depeng¹,Wang Rui¹

Affiliation:

1. Key Laboratory of Preclinical Study for New Drugs of Gansu Province, School of Basic Medical Sciences, and Institute of Biochemistry and Molecular Biology, Lanzhou University, Lanzhou, 730000, P. R. China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm400195y

Reference92 articles.

1. The Endogenous Opioid System and Clinical Pain Management

2. Opioid Receptors and their Ligands

3. Opioid receptor targeting ligands for pain management: a review and update

4. A potent and selective endogenous agonist for the µ-opiate receptor

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