Structure-Based Design, Synthesis, and Biochemical and Pharmacological Characterization of Novel Salvinorin A Analogues as Active State Probes of the κ-Opioid Receptor-Reference-Cited by-同舟云学术

Structure-Based Design, Synthesis, and Biochemical and Pharmacological Characterization of Novel Salvinorin A Analogues as Active State Probes of the κ-Opioid Receptor

Published:2009-07-06 Issue:29 Volume:48 Page:6898-6908
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Yan Feng¹,Bikbulatov Ruslan V.²,Mocanu Viorel³⁴,Dicheva Nedyalka³,Parker Carol E.³,Wetsel William C.⁵,Mosier Philip D.⁶,Westkaemper Richard B.⁶,Allen John A.¹,Zjawiony Jordan K.²⁷,Roth Bryan L.¹

Affiliation:

1. Department of Pharmacology

2. Department of Pharmacognosy, School of Pharmacy, University of Mississippi, University, Mississippi 38677

3. UNC-Duke Proteomics Center

4. Deceased.

5. Department of Cell Biology, Duke University Medical Center, Durham, North Carolina 27710

6. Department of Medicinal Chemistry, Virginia Commonwealth University, Richmond, Virginia 23298

7. National Center for Natural Products Research, Research Institute of Pharmaceutical Sciences, School of Pharmacy, University of Mississippi, University, Mississippi 38677

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/bi900605n

Reference42 articles.

1. Salvinorin, a new trans-neoclerodane diterpene from Salvia divinorum(Labiatae)

2. Divinorin A, a psychotropic terpenoid, and divinorin B from the hallucinogenic Mexican mint, Salvia divinorum

3. Salvinorin A: A potent naturally occurring nonnitrogenous opioid selective agonist

4. Antinociceptive and Hypothermic Effects of Salvinorin A Are Abolished in a Novel Strain of κ-Opioid Receptor-1 Knockout Mice

5. Salvinorin A: the ‘magic mint’ hallucinogen finds a molecular target in the kappa opioid receptor

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