New Nitrogen Containing Substituents at the Indole-2-carboxamide Yield High Potent and Broad Spectrum Indolylarylsulfone HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors-Reference-Cited by-同舟云学术

New Nitrogen Containing Substituents at the Indole-2-carboxamide Yield High Potent and Broad Spectrum Indolylarylsulfone HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors

Published:2012-07-06 Issue:14 Volume:55 Page:6634-6638
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

La Regina Giuseppe¹,Coluccia Antonio¹,Brancale Andrea²,Piscitelli Francesco¹,Famiglini Valeria¹,Cosconati Sandro³,Maga Giovanni⁴,Samuele Alberta⁴,Gonzalez Emmanuel⁵,Clotet Bonaventura⁵,Schols Dominique⁶,Esté José A.⁵,Novellino Ettore⁷,Silvestri Romano¹

Affiliation:

1. Istituto Pasteur - Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, Piazzale Aldo Moro 5, I-00185 Roma, Italy

2. Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff, CF10 3NB, U.K., Istituto di Chimica Biomolecolare, CNR, Piazzale Aldo Moro 5, I-00185 Roma, Italy

3. Dipartimento di Scienze Ambientali, Seconda Università di Napoli, Via Vivaldi 43, 81100 Caserta, Italy

4. Institute of Molecular Genetics IGM-CNR, National Research Council, via Abbiategrasso 207, I-27100 Pavia, Italy

5. IrsiCaixa, Hospital Universitari Germans Trias i Pujol, Universitat Autonoma de Barcelona, 08916 Badalona, Spain

6. Rega Institute for Medical Research, Katholieke Universiteit Leuven, B-3000 Leuven, Belgium

7. Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, Via Domenico Montesano 49, I-80131, Napoli, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300477h

Reference18 articles.

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