Lysergamides of Isomeric 2,4-Dimethylazetidines Map the Binding Orientation of the Diethylamide Moiety in the Potent Hallucinogenic Agent N,N-Diethyllysergamide (LSD)-Reference-Cited by-同舟云学术

Lysergamides of Isomeric 2,4-Dimethylazetidines Map the Binding Orientation of the Diethylamide Moiety in the Potent Hallucinogenic Agent N,N-Diethyllysergamide (LSD)

Published:2002-09-01 Issue:19 Volume:45 Page:4344-4349
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nichols David E.¹,Frescas Stewart¹,Marona-Lewicka Danuta¹,Kurrasch-Orbaugh Deborah M.¹

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, School of Pharmacy and Pharmacal Sciences, Purdue University, West Lafayette, Indiana 47907

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020153s

Reference26 articles.

1. Drug discrimination and receptor binding studies of N-isopropyl lysergamide derivatives

2. Stereoselective LSD-like activity in d-lysergic acid amides of R- and S-2-aminobutane

3. Complex stimulus properties of LSD: a drug discrimination study with α2-adrenoceptor agonists and antagonists

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