Synthesis and Structure−Activity Relationships of β- and α-Piperidine Sulfone Hydroxamic Acid Matrix Metalloproteinase Inhibitors with Oral Antitumor Efficacy-Reference-Cited by-同舟云学术

Synthesis and Structure−Activity Relationships of β- and α-Piperidine Sulfone Hydroxamic Acid Matrix Metalloproteinase Inhibitors with Oral Antitumor Efficacy

Published:2005-09-21 Issue:21 Volume:48 Page:6713-6730
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Becker Daniel P.¹,Villamil Clara I.¹,Barta Thomas E.¹,Bedell Louis J.¹,Boehm Terri L.¹,DeCrescenzo Gary A.¹,Freskos John N.¹,Getman Daniel P.¹,Hockerman Susan¹,Heintz Robert¹,Howard Susan Carol¹,Li Madeleine H.¹,McDonald Joseph J.¹,Carron Chris P.¹,Funckes-Shippy Chris L.¹,Mehta Pramod P.¹,Munie Grace E.¹,Swearingen Craig A.¹

Affiliation:

1. Pfizer Research, 4901 Searle Parkway, Skokie, Illinois 60077, and Pfizer Research, 700 Chesterfield Village Parkway, St. Louis, Missouri 63198

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0500875

Reference42 articles.

1. Matrix metalloproteinases: a tail of a frog that became a prince

2. Matrix Metalloproteinases

3. The Design, Structure, and Therapeutic Application of Matrix Metalloproteinase Inhibitors

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