Effects of Heterocyclic Aromatic Substituents on Binding Affinities at Two Distinct Sites of Somatostatin Receptors. Correlation with the Electrostatic Potential of the Substituents-Reference-Cited by-同舟云学术

Effects of Heterocyclic Aromatic Substituents on Binding Affinities at Two Distinct Sites of Somatostatin Receptors. Correlation with the Electrostatic Potential of the Substituents

Published:2003-04-15 Issue:10 Volume:46 Page:1858-1869
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Prasad Vidya¹,Birzin Elizabeth T.¹,McVaugh Cheryl T.¹,van Rijn Rachel D.¹,Rohrer Susan P.¹,Chicchi Gary¹,Underwood Dennis J.¹,Thornton Edward R.¹,Smith Amos B.¹,Hirschmann Ralph¹

Affiliation:

1. Department of Chemistry, University of Pennsylvania, Philadelphia, Pennsylvania 19104, Merck Research Laboratories, Rahway, New Jersey 07065, and DuPont Pharmaceutical Company, Wilmington, Delaware 19880

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0205088

Reference58 articles.

1. De novo design and synthesis of somatostatin non-peptide peptidomimetics utilizing .beta.-D-glucose as a novel scaffolding

2. On the origins of the DNA sequence selectivity of mitomycin monoalkylation transformations

3. Modulation of Receptor and Receptor Subtype Affinities Using Diastereomeric and Enantiomeric Monosaccharide Scaffolds as a Means to Structural and Biological Diversity. A New Route to Ether Synthesis

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