1. Selected reviews on β-turn mimics: (a) Rose, G. D.; Gierasch, L. M.; Smith, J. A. InAdvances in Protein Chemistry; Anfinsen, C. B., Edsall, J. T., Richards, F. M., Eds.; Academic: Orlando, FL, 1985; Vol. 37, pp 1−109. (b) Giannis, A.; Kolter, T.Angew. Chem., Int. Ed. Engl.1993,32, 1244−1267. (c) Nagai, U.; Sato, K.; Nakamura, R.; Kato, R.Tetrahedron1993,49, 3577−3592. (d) Olson, G. L.; Bolin, D. R.; Bonner, M. P.; Bös, M.; Cook, C. M.; Fry, D. C.; Graves, B. J.; Hatada, M.; Hill, D. E.; Kahn, M.; Madison, V. S.; Rusiecki, V. K.; Sarabu, R.; Sepinwall, J.; Vincent, G. P.; Voss, M. E.J. Med. Chem.1993,36, 3039−3049. (e) Mueller, G.Angew. Chem., Int. Ed. Engl.1997,35, 2767−2769. (f) MacDonald, M.; Aubé, J.Curr. Org. Chem.2001,5, 417−438. (g) Hanessian, S.; McNaughton-Smith, G.; Lombart, H.G.; Lubell, W. D.Tetrahedron1997,53, 12789−12854. (h) Burgess, K.Acc. Chem. Res.2001,34, 826−835. (i) Nubbemeyer, U.Top. Curr. Chem.2001,216, 125−196. (j) Souers, A. J.; Ellman, J. A.Tetrahedron2001,57, 7431−7448. (k) Eguchi, M.; Kahn, M.Mini-Rev. Med. Chem.2002,2, 447−462. (l) Hruby, V. J.Nat. Rev. Drug Discovery2002,1, 847−858. (m) Suat Kee, K.; Jois, S. D. S.Curr. Pharm. Des.2003,9, 1209−1224. (n) Ahn, J.M.; Boyle, N. A.; MacDonald, M. T.; Janda, K. D.Mini-Rev. Med. Chem.2002,2, 463−473.
2. Solid-Phase SN2 Macrocyclization Reactions To Form β-Turn Mimics
3. Solid-Phase SNAr Macrocyclizations To Give Turn-Extended-Turn Peptidomimetics