Novel N-Arylpyrazolo[3,2-c]-Based Ligands for the Glucocorticoid Receptor: Receptor Binding and in Vivo Activity-Reference-Cited by-同舟云学术

Novel N-Arylpyrazolo[3,2-c]-Based Ligands for the Glucocorticoid Receptor: Receptor Binding and in Vivo Activity

Published:2004-04-02 Issue:10 Volume:47 Page:2441-2452
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ali Amjad¹,Thompson Christopher F.¹,Balkovec James M.¹,Graham Donald W.¹,Hammond Milton L.¹,Quraishi Nazia¹,Tata James R.¹,Einstein Monica¹,Ge Lan¹,Harris Georgianna¹,Kelly Terri M.¹,Mazur Paul¹,Pandit Shilpa¹,Santoro Joseph¹,Sitlani Ayesha¹,Wang Chuanlin¹,Williamson Joanne¹,Miller Douglas K.¹,Thompson Chris M.¹,Zaller Dennis M.¹,Forrest Michael J.¹,Carballo-Jane Ester¹,Luell Silvi¹

Affiliation:

1. Departments of Medicinal Chemistry, Metabolic Disorders, Immunonology, and Pharmacology, Merck Research Laboratories, P.O. Box 2000, Rahway, New Jersey 07065

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030585i

Reference33 articles.

1. 16-Methylated Steroids. IV. 6,16α-Dimethyl-▵6-Hydrocortisone and Related Compounds

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