Novel Highly Potent and Selective Nonsteroidal Aromatase Inhibitors: Synthesis, Biological Evaluation and Structure−Activity Relationships Investigation-Reference-Cited by-同舟云学术

Novel Highly Potent and Selective Nonsteroidal Aromatase Inhibitors: Synthesis, Biological Evaluation and Structure−Activity Relationships Investigation

Published:2010-06-22 Issue:14 Volume:53 Page:5347-5351
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gobbi Silvia¹,Zimmer Christina²,Belluti Federica¹,Rampa Angela¹,Hartmann Rolf W.²,Recanatini Maurizio¹,Bisi Alessandra¹

Affiliation:

1. Department of Pharmaceutical Sciences, University of Bologna, Via Belmeloro 6, I-40126 Bologna, Italy

2. Pharmaceutical and Medicinal Chemistry, Saarland University, P.O. Box 151150, & Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), D-66041 Saarbrücken, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100319h

Reference30 articles.

1. Cancer Facts & Figures 2009;American Cancer Society:Atlanta, GA,2010.

2. In situestrogen production and its regulation in human breast carcinoma: From endocrinology to intracrinology

3. History of Aromatase: Saga of an Important Biological Mediator and Therapeutic Target

4. First-line endocrine treatment of breast cancer: aromatase inhibitor or antioestrogen?

5. Aromatase Inhibitors in Early Hormone Receptor-Positive Breast Cancer

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