Development of a Practical Synthesis of Functionalized Azaxanthene-Derived Nonsteroidal Glucocorticoid Receptor Modulators-Reference-Cited by-同舟云学术

Development of a Practical Synthesis of Functionalized Azaxanthene-Derived Nonsteroidal Glucocorticoid Receptor Modulators

Published:2016-05-12 Issue:5 Volume:20 Page:921-933
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Conlon David A.,Natalie Kenneth J.,Cuniere Nicolas,Razler Thomas M.,Zhu Jason,de Mas Nuria,Tymonko Steven,Fraunhoffer Kenneth J.,Sortore Eric,Rosso Victor W.,Xu Zhongmin,Adams Monica L.,Patel Anisha,Huang Jun,Gong Hua¹,Weinstein David S.¹,Quiroz Fernando,Chen Doris C.

Affiliation:

1. Research and Development, Bristol-Myers Squibb, Princeton, New Jersey 08543-4000, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.6b00035

Reference40 articles.

1. Selective glucocorticoid receptor agonists (SEGRAs): Novel ligands with an improved therapeutic index

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4. Mechanisms involved in the side effects of glucocorticoids

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