Effect of Temperature and Solvent of Solvent-Mediated Polymorph Transformation on ASP3026 Polymorphs and Scale-up-Reference-Cited by-同舟云学术

Effect of Temperature and Solvent of Solvent-Mediated Polymorph Transformation on ASP3026 Polymorphs and Scale-up

Published:2016-04-28 Issue:5 Volume:20 Page:970-976
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Takeguchi Kazuhiro¹²,Obitsu Kazuyoshi¹,Hirasawa Shun¹,Orii Ryoki¹,Ieda Shigeru³,Okada Minoru¹,Takiyama Hiroshi²

Affiliation:

1. Technology Process Chemistry Laboratories, Astellas Pharma Inc., 160-2 Akahama, Takahagi, Ibaraki 318-0001, Japan

2. Department of Chemical Engineering, Tokyo University of Agriculture and Technology, 2-24-16, Naka-cho, Koganei, Tokyo 184-8588, Japan

3. Astellas Pharma Tech Co., Ltd., 160-2 Akahama, Takahagi, Ibaraki 318-0001, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.6b00068

Reference14 articles.

1. Crystal structures of drugs: advances in determination, prediction and engineering

2. Pharmaceutical Applications of Polymorphism

3. Kondoh, Y.; Hkubo, K.; Kuromitsu, S.; Shindo, N.; Soga, T.; Furutani, T.; Shimada, I.; Matsuya, T.; Kurosawa, K.; Kamikawa, A.; Mano, H.PCT Int. Appl. Di(arylamino)aryl Compound.WO 2009008371Al, 2009.

4. Shimada, I.; Hirakura, Y.; Yamazaki, K.; Takeguchi, K.; Ueda, N.PCT Int. Appl. Crystals of Di(arylamino)aryl Compound. WO2011145548A1, 2011.

Cited by 21 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Cocrystal of Naringenin and Norfloxacin: Crystal Transformation, Solubility, and Antibacterial and Anticancer Activities;Crystal Growth & Design;2024-05-25

2. Solvent-Mediated Hetero/Homo-Phase Crystallization of Copper Nanoclusters and Superatomic Kernel-Related NIR Phosphorescence;Journal of the American Chemical Society;2024-04-09

3. Mechanistic Study on the Effect of Solvents on Polymorphic Transformation of Aripiprazole by Solvent Property Parameters and Molecular Dynamics Simulation;Crystal Growth & Design;2024-03-18

4. Insight into the Structure and Property Diversity of Four Nicorandil Oxalate Salt Polymorphs Based on Experiments and Quantum Chemistry Study;Crystal Growth & Design;2024-01-13

5. Hydration Mechanism and Its Effect on the Solubility of Aripiprazole;Pharmaceutical Research;2023-10-13