Enantioselective Synthesis of the Chiral Pyrrolidine Fragment of Upadacitinib <i>via</i> Chiral Auxiliary Directed Diastereoselective 1,3-Dipolar Cycloaddition-Reference-Cited by-同舟云学术

Enantioselective Synthesis of the Chiral Pyrrolidine Fragment of Upadacitinib via Chiral Auxiliary Directed Diastereoselective 1,3-Dipolar Cycloaddition

Published:2022-05-20 Issue:6 Volume:26 Page:1794-1802
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Sampath Magesh¹,Jayaraman Sembian Ruso¹,Eda Vishnuvardhan Reddy¹,Potham Rajendar¹,Budhdev Rajeev Rehani²,Sen Saikat¹,Bandichhor Rakeshwar²^ORCID,Oruganti Srinivas¹^ORCID

Affiliation:

1. Dr. Reddy’s Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, Telangana, India

2. Integrated Product Development Organization, Dr. Reddy’s Laboratories, Bachupally, Qutbullapur, Hyderabad 500 090, Telangana, India

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.1c00454

Reference38 articles.

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