Improved Synthetic Process of Baloxavir Marboxil Intermediate 3-Benzyloxy-4-oxo-4<i>H</i>-pyran-2-carboxylic Acid-Reference-Cited by-同舟云学术

Improved Synthetic Process of Baloxavir Marboxil Intermediate 3-Benzyloxy-4-oxo-4H-pyran-2-carboxylic Acid

Published:2023-06-02 Issue:6 Volume:27 Page:1015-1026
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Huang Kongcheng¹²^ORCID,Lu Jianwu³²^ORCID,Wang Xiaoxu²,Shi Yinfei²,Yang Kaimike⁴,Yuan Shun²,Wang Yinquan²,Sun Han²,Liu Yuebin²,Sun Xun³^ORCID,Wu Taizhi²^ORCID

Affiliation:

1. School of Chemistry and Chemical Engineering, Shanghai University of Engineering Science, 333 Longteng Road, Shanghai 201620, China

2. State Key Lab of New Drug & Pharmaceutical Process, Shanghai Institute of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, China

3. Department of Natural Medicine, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai 201203, China

4. Wuhan Britain-China Senior High School, 10 Gutian Ce Road, Wuhan 430061, China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.2c00387

Reference35 articles.

1. Baloxavir Marboxil: The First Cap-Dependent Endonuclease Inhibitor for the Treatment of Influenza

2. Dolutegravir for the treatment of HIV

3. Baloxavir marboxil: the new influenza drug on the market

4. World Health Organization. Influenza (Seasonal). Https://www.who.int/news-room/fact-sheets/detail/influenza-(seasonal) (accessed April 14, 2023).

5. Johns, B. A.; Weatherhead, J. G. Chemical Compounds. WO 2010011815 A1, 2010.

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