Two Approaches to the Chemical Development and Large-Scale Preparation of a Pyrimidyl Tetrazole Intermediate-Reference-Cited by-同舟云学术

Two Approaches to the Chemical Development and Large-Scale Preparation of a Pyrimidyl Tetrazole Intermediate

Published:2016-06-08 Issue:6 Volume:20 Page:1075-1087
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Mullens Peter¹,Cleator Ed¹,McLaughlin Mark²,Bishop Brian¹,Edwards John¹,Goodyear Adrian¹,Andreani Teresa²,Jin Yan²,Kong Jongrock²,Li Hongmei²,Williams Michael²,Zacuto Michael²

Affiliation:

1. Department of Process & Analytical Chemistry, Merck, Sharp and Dohme Ltd., Hertford Road, Hoddesdon, EN11 9BU, U.K.

2. Department of Process & Analytical Chemistry, Merck Research Laboratories, Merck & Co., Inc., Rahway, New Jersey 07065, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.6b00136

Reference25 articles.

1. Synthesis of 1-substituted tetrazoles via the acid-catalyzed [3+2] cycloaddition between isocyanides and trimethylsilyl azide

2. The Promise and Challenge of Iron-Catalyzed Cross Coupling

3. Preparation of Carboxylic Acids from Aldehydes (Including Hydroxylated Benzaldehydes) by Oxidation with Chlorite.

4. Model studies for the synthesis of quassinoids. 1. Construction of the BCE ring system

5. Synthetic studies toward verrucarol. 2. Synthesis of the AB ring system

Cited by 18 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Covalent Organic Frameworks as a Versatile Platform for Iron‐Catalyzed sp³ C−H Activation and Cross‐Coupling via Decarboxylative Oxidation;European Journal of Inorganic Chemistry;2024-03

2. Anwendung von Organometallkatalysatoren in der API-Synthese;Organometallik in der Prozesschemie;2024

3. Cu-Mediated Ullmann-Type Cross-Coupling and Industrial Applications in Route Design, Process Development, and Scale-up of Pharmaceutical and Agrochemical Processes;Organic Process Research & Development;2022-05-24

4. Iron Catalyzed C–C-Bond Formation: From Canonical Cross Coupling to a Quest for New Reactivity;Bulletin of the Chemical Society of Japan;2021-02-15

5. Discussion Addendum for: 4‐Nonylbenzoic Acid;Organic Syntheses;2020-04-29