A Simple and Commercially Viable Process for Improved Yields of Metopimazine, a Dopamine D2-Receptor Antagonist-Reference-Cited by-同舟云学术

A Simple and Commercially Viable Process for Improved Yields of Metopimazine, a Dopamine D2-Receptor Antagonist

Published:2017-05-11 Issue:5 Volume:21 Page:720-731
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Karicherla Venumanikanta¹,Phani Kumar¹,Bodireddy Mohan Reddy¹,Prashanth Kumar Babu¹,Gajula Madhusudana Rao¹,Pramod Kumar¹^ORCID

Affiliation:

1. Chemical Research Division, API R&D Centre, Micro Labs Ltd., Plot No.43-45, KIADB Industrial Area, Fourth Phase, Bommasandra-Jigani Link Road, Bommasandra, Bangalore, Karnataka 560 105, India

Funder

Micro Labs Limited

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.7b00052

Reference29 articles.

1. Antiemetics for Cancer Chemotherapy-Induced Nausea and Vomiting

2. Control of Chemotherapy-Induced Emesis

3. Randomized, double-blind comparison of ondansetron versus ondansetron plus metopimazine as antiemetic prophylaxis during platinum-based chemotherapy in patients with cancer.

4. Ann. Drug Data Rep.;Prous, J. R.; Vedrilla, D., Eds.Drugs of Today:Barcelona, Spain, 1971.1, 293

5. Antiemetic specificity of dopamine antagonists

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