Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor-Reference-Cited by-同舟云学术

Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor

Published:2019-10-18 Issue:11 Volume:23 Page:2482-2498
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Fraunhoffer Kenneth J.¹^ORCID,DelMonte Albert J.¹^ORCID,Beutner Gregory L.¹^ORCID,Bultman Michael S.¹^ORCID,Camacho Kathryn¹,Cohen Benjamin¹^ORCID,Dixon Darryl D.¹^ORCID,Fan Yu¹,Fanfair Dayne¹,Freitag Adam J.¹,Glace Andrew W.¹,Gonzalez-Bobes Francisco¹^ORCID,Gujjar Manjunath²,Haley Matthew W.¹,Hickey Matthew R.¹,Ho Jeanne¹,Iyer Vidya¹,Maity Prantik²,Patel Sunil¹,Rosso Victor W.¹,Schmidt Michael A.¹^ORCID,Stevens Jason M.¹^ORCID,Tan Yichen¹,Wilbert Christopher¹,Young Ian S.¹^ORCID,Yu Miao¹^ORCID

Affiliation:

1. Chemical and Synthetic Development, Bristol-Myers Squibb Global Product Development and Supply, One Squibb Drive, P.O. Box 191, New Brunswick, New Jersey 08903-0191, United States

2. Chemical and Synthetic Development, Biocon Bristol-Myers Squibb Research and Development Center, Biocon Park, Jigani Link Road, Bommasandra IV, Bangalore 560099, India

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.9b00359

Reference30 articles.

1. National Cancer Institute Cancer Statistics. https://www.cancer.gov/about-cancer/understanding/statistics (accessed Nov 21, 2017).

2. Why tumours eat tryptophan

3. Immune-modulating enzyme indoleamine 2,3-dioxygenase is effectively inhibited by targeting its apo-form

4. Beck, H. P.; Jaen, J. C.; Osipov, M.; Powers, J. P.; Reilly, M. K.; Shunatona, H. P.; Walker, J. R.; Zibinsky, M.; Balog, J. A.; Williams, D. K.; Markwalder, J. A.; Cherney, E.; Shan, W.; Huang, A. Immunoregulatory Agents. WO2016073770A1, May 12, 2016.

5. Lanthanoids in organic synthesis. 5. Selective reductions of ketones in the presence of aldehydes

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