Practical Synthesis of Chiral 3-(Hydroxyiminomethyl)adipic Acid, a Key Intermediate of the ROR-γ Inhibitor JTE-151, via Crystallization-Induced Dynamic Resolution-Reference-Cited by-同舟云学术

Practical Synthesis of Chiral 3-(Hydroxyiminomethyl)adipic Acid, a Key Intermediate of the ROR-γ Inhibitor JTE-151, via Crystallization-Induced Dynamic Resolution

Published:2023-11-20 Issue:12 Volume:27 Page:2355-2364
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Takiguchi Hiromu¹^ORCID,Watanabe Takashi¹,Ogo Takashi¹,Ishibashi Hideaki¹,Yokota Katsuyuki¹,Obika Shingo¹,Inaba Takashi¹

Affiliation:

1. Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1 Murasaki-cho, Takatsuki, Osaka 569-1125, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.3c00320

Reference25 articles.

1. Retinoic Acid Receptor-Related Orphan Receptor γt (RORγt) Agonists as Potential Small Molecule Therapeutics for Cancer Immunotherapy

2. Modulators of the Nuclear Receptor Retinoic Acid Receptor-Related Orphan Receptor-γ (RORγ or RORc)

3. Maeba, T.; Maeda, K.; Kotoku, M.; Hirata, K.; Seki, N.; Yamanaka, H.; Sakai, T.; Hirashima, S.; Obika, S.; Shiozaki, M.; Yokota, M. Amide compound and pharmaceutical application therefor. WO Patent WO2012/147916A1, 2012.

4. 1112. Derivatives of 6-aminopenicillanic acid. Part VI. Penicillins from 3- and 5-phenylisoxazole-4-carboxylic acids and their alkyl and halogen derivatives

5. Recent Developments in the Synthesis and Reactivity of Isoxazoles: Metal Catalysis and Beyond

Cited by 1 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Practical Manufacturing Process for Baloxavir Marboxil: Effective Selection and Replacement of Protective Group toward Enhancement of Crystallization-Induced Diastereomer Transformation;Organic Process Research & Development;2024-04-04