Optimization and Scale-Up of a Continuous Flow Synthesis of Dapagliflozin-Reference-Cited by-同舟云学术

Optimization and Scale-Up of a Continuous Flow Synthesis of Dapagliflozin

Published:2023-02-08 Issue: Volume: Page:
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Wang Chunchao¹,Xuan Boxin¹,Huang Cheng¹,Yao Jingchun²,Wu Chengjun¹²,Sun Tiemin¹^ORCID

Affiliation:

1. Key Laboratory of Structure-Based Drug Design and Discovery, Shenyang Pharmaceutical University, Ministry of Education. Shenyang 110016, P.R. China

2. State Key Laboratory of Generic Manufacture Technology of Chinese Traditional Medicine, Lunan Pharmaceutical Group Co. LTD., Linyi, 276005, China

Funder

Department of Education of Liaoning Province

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.2c00389

Reference30 articles.

1. Discovery of Dapagliflozin: A Potent, Selective Renal Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitor for the Treatment of Type 2 Diabetes

2. Dapagliflozin: A Review in Type 2 Diabetes

3. Applicability of US Food and Drug Administration Labeling for Dapagliflozin to Patients With Heart Failure With Reduced Ejection Fraction in US Clinical Practice

4. Effects of Dapagliflozin in Stage 4 Chronic Kidney Disease

5. Molecular Characteristics of Na+-coupled Glucose Transporters in Adult and Embryonic Rat Kidney

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