Direct Synthesis of a PDE4 Inhibitor by Using Pd–Cu-Catalyzed C–H/C–Br Coupling of Benzoxazole with a Heteroaryl Bromide-Reference-Cited by-同舟云学术

Direct Synthesis of a PDE4 Inhibitor by Using Pd–Cu-Catalyzed C–H/C–Br Coupling of Benzoxazole with a Heteroaryl Bromide

Published:2016-05-18 Issue:6 Volume:20 Page:1053-1058
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Kuroda Kiichi¹,Tsuyumine Shinjiro¹,Kodama Tomohiro¹

Affiliation:

1. Process Chemistry Research and Development Laboratories, Technology Research & Development Division and ‡DSP Cancer Institute, Sumitomo Dainippon Pharma Company, Ltd., 3-1-98 Kasugade-naka, Konohana-ku, Osaka 554-0022, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.6b00106

Reference23 articles.

1. aIshikawa, J.; Saito, K.; Ohe, N.; Kobayashi, K.PCT int. Appl. WO2010/137349 A1.

2. bPatent pending.

3. Novel fluorescent quater- and quinquifurans: Syntheses and photophysical properties

4. Recent advances in the total syntheses of oxazole-containing natural products

5. Palladium-Catalyzed Cross-Coupling Reactions in Total Synthesis

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