Practical Synthesis of a S1P Receptor 1 Agonist via a Guareschi–Thorpe Reaction
Author:
Affiliation:
1. Chemistry Process R&D, Actelion Pharmaceuticals Ltd., Gewerbestrasse 16, CH-4123 Allschwil, Switzerland
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.6b00210
Reference28 articles.
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3. Practical and Scalable Synthesis of S1P1 Receptor Agonist ACT-209905
4. Synthesis of 2,6-di(pyrazol-1-yl)-4-bromomethylpyridine, and its conversion to other 2,6-di(pyrazol-1-yl)pyridines substituted at the pyridine ring
5. Markley, L. D.; Soper, J. M.US 4474602, 1984.
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