Investigating Scale-Up and Further Applications of DABAL-Me3 Promoted Amide Synthesis-Reference-Cited by-同舟云学术

Investigating Scale-Up and Further Applications of DABAL-Me3 Promoted Amide Synthesis

Published:2015-06-24 Issue:7 Volume:19 Page:831-840
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Lee Darren S.¹,Amara Zacharias¹,Poliakoff Martyn¹,Harman Thomas²,Reid Gary²,Rhodes Barrie²,Brough Steve³,McInally Thomas¹,Woodward Simon¹

Affiliation:

1. School of Chemistry, University of Nottingham, University Park, Nottingham, NG7 2RD, United Kingdom

2. Aesica Pharmaceuticals Ltd., Quorum Business Park, Benton Lane, Newcastle upon Tyne, NE12 8BS, United Kingdom

3. Key Organics Ltd., Highfield Road Industrial Estate, Camelford, Cornwall, PL32 9RA, United Kingdom

Funder

University Of Nottingham

Engineering and Physical Sciences Research Council

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.5b00101

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5. bKhan, T.; Josien, H.; McKittrick, B.; Vaccaro, H.; Bara, T.; Caldwell, J.; Heap, C. R.; Giess, W. B.; Mitra, S.; Zych, A. J.Preparation of N3-substituted iminopyrimidinones as renin inhibitors, compositions, and their use. WO 2013/142396 A1, 2013.

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