Kilogram-Scale Preparation of an Aminopyrazole Building Block via Copper-Catalyzed Aryl Amidation-Reference-Cited by-同舟云学术

Kilogram-Scale Preparation of an Aminopyrazole Building Block via Copper-Catalyzed Aryl Amidation

Published:2021-04-06 Issue:4 Volume:25 Page:1065-1073
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Baldwin Aaron F.¹,Caporello Michaella A.²,Chen Guoyong³,Goetz Adam E.²^ORCID,Hu Weifeng³,Jin Chengfeng³,Knopf Kevin M.²,Li Zhifeng³,Lu Cuong V.²,Monfette Sebastien²,Puchlopek-Dermenci Angela L. A.²,Shi Feng³

Affiliation:

1. Analytical Research and Development, Pfizer Worldwide Research and Development, Groton Laboratories, Eastern Point Road, Groton, Connecticut 06340, United States

2. Chemical Research and Development, Pfizer Worldwide Research and Development, Groton Laboratories, Eastern Point Road, Groton, Connecticut 06340, United States

3. Shanghai STA Pharmaceutical R&D Co. Ltd., #90 Delin Road, WaiGaoQiao Free Trade Zone, Shanghai 200131, China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.1c00066

Reference76 articles.

1. Synthesis of Anilines

2. Advancement in methodologies for reduction of nitroarenes

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5. Risk Assessment of Potentially Genotoxic Impurities within the Framework of Quality by Design

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