A Concise and Efficient Synthesis of Dapagliflozin-Reference-Cited by-同舟云学术

A Concise and Efficient Synthesis of Dapagliflozin

Published:2019-06-27 Issue:7 Volume:23 Page:1458-1461
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Yu Jun¹^ORCID,Cao Ying¹,Yu HaiZhou¹,Wang JinJia¹

Affiliation:

1. The Research Academy of Jiangsu Hansoh Pharmaceutical Co., LTD, Dongjin Road, Huaguoshan Avenue, Lianyungang, Jiangsu 222069, P. R. China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.9b00141

Reference18 articles.

1. Discovery of Dapagliflozin: A Potent, Selective Renal Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitor for the Treatment of Type 2 Diabetes

2. Ellsworth, B.; Washburn, W. N.; Sher, P. M.; Wu, G.; Meng, W. C-Aryl Glucoside SGLT2 Inhibitors and Method. US 6515117 B2, 2003.

3. Deshpande, P. P.; Ellsworth, B. A.; Singh, J.; Denzel, T.; Lai, C.; Crispino, G.; Randazzo, M. E.; Gougoutas, J. Z. Methods of Producing C-Aryl Glucoside SGLT2 Inhibitors. US 7375213 B2, 2008.

4. Glycosyl Cross-Coupling of Anomeric Nucleophiles: Scope, Mechanism, and Applications in the Synthesis of Aryl C-Glycosides

5. Synthetic routes to higher-carbon sugars. Reaction of lactones with 2-lithio-,3-dithiane

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