1. The benzodiazepine story
2. (a)Gosmini, R. L. M.; Mirguet, O. Benzodiazepine derivatives as bromodomain inhibitor and their preparation and use in the treatment of cancer, chronic autoimmune and inflammatory disease PCT WO 2,011,054,553 A1, 12 May 2011
3. (b)Burns, C.; Garnier, J-M.; Sharp, P. P.; Feutrill, J.; Cuzzupe, A. Preparation of benzodiazepine derivatives as bromodomain inhibitors PCT WO 2,017,020,086 A1, 9 February 2017.
4. Siegel, S.; Baeurle, S.; Cleve, A.; Haendler, B.; Fernandez-Montalvan, A. E.; Moenning, U.; Krause, S.; Lejeune, P.; Busemann, M.; Kuhnke, J. Bicyclo 2,3-benzodiazepines and spirocyclically substituted 2,3-benzodiazepines PCT Int. Appl. WO 2,014,128,067 A1, 28 August 2014.