Development of a Multikilogram Scale Synthesis of a TRPV1 Antagonist
Author:
Affiliation:
1. Department of Process Chemistry, Merck & Co., Inc., Rahway, New Jersey 07065, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.5b00388
Reference28 articles.
1. The vanilloid receptor TRPV1: 10 years from channel cloning to antagonist proof-of-concept
2. Recent Progress in the Development of Selective TRPV1 Antagonists for Pain
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5. Targeting Pain-evoking Transient Receptor Potential Channels for the Treatment of Pain
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