Development of a Synthesis of a 2,3-Disubstituted 4,7-Diazaindole Including Large-Scale Application of CH3Li/TiCl4-Mediated Methylation of an Enolizable Ketone-Reference-Cited by-同舟云学术

Development of a Synthesis of a 2,3-Disubstituted 4,7-Diazaindole Including Large-Scale Application of CH3Li/TiCl4-Mediated Methylation of an Enolizable Ketone

Published:2015-06-26 Issue:7 Volume:19 Page:806-811
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Weiberth Franz J.¹,Gill Harpal S.¹,Lee George E.¹,Ngo Duc P.¹,Shrimp Frederick L.¹,Chen Xuemin¹,D’Netto Geoffrey¹,Jackson Bryan R.¹,Jiang Ying¹,Kumar Narendra¹,Roberts Frederick¹,Zlotnikov Evgeny¹

Affiliation:

1. Synthesis Development, Sanofi U.S. R&D, 153 Second Avenue, Waltham, Massachusetts 02451, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op5003769

Reference18 articles.

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2. Iron-Catalyzed Cross-Coupling Reactions

3. Selective Iron-Catalyzed Cross-Coupling Reactions of Grignard Reagents with Enol Triflates, Acid Chlorides, and Dichloroarenes

4. Cyclisation par amination intramoléculaire dans la série de la pyrazine.

5. Lee, G. E.; Shrimp, F. L., II; Weiberth, F. J.PCT Int. Appl.WO 2010/107969A1, 2010.

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