The Glutamate Receptor GluR5 Agonist (S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid and the 8-Methyl Analogue: Synthesis, Molecular Pharmacology, and Biostructural Characterization†PDB ID: 2WKY.
Author:
Affiliation:
1. Department of Medicinal Chemistry
2. Department of Pharmacology and Pharmacotherapy
3. Faculty of Pharmaceutical Sciences, University of Copenhagen, 2 Universitetsparken, DK-2100 Copenhagen, Denmark
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm900565c
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1. Ligands for Glutamate Receptors: Design and Therapeutic Prospects
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3. Glutamate in CNS disorders as a target for drug development: an update
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