Discovery of a Fluoroindolo[2,3-a]carbazole Clinical Candidate with Broad Spectrum Antitumor Activity in Preclinical Tumor Models Superior to the Marketed Oncology Drug, CPT-11-Reference-Cited by-同舟云学术

Discovery of a Fluoroindolo[2,3-a]carbazole Clinical Candidate with Broad Spectrum Antitumor Activity in Preclinical Tumor Models Superior to the Marketed Oncology Drug, CPT-11

Published:2005-02-16 Issue:7 Volume:48 Page:2258-2261
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Saulnier Mark G.¹,Balasubramanian Balu N.¹,Long Byron H.¹,Frennesson David B.¹,Ruediger Edward¹,Zimmermann Kurt¹,Eummer Jeffrey T.¹,St. Laurent Denis R.¹,Stoffan Karen M.¹,Naidu B. Narasimhulu¹,Mahler Mikael¹,Beaulieu Francis¹,Bachand Carol¹,Lee Frank Y.¹,Fairchild Craig R.¹,Stadnick Linda K.¹,Rose William C.¹,Solomon Carola¹,Wong Henry¹,Martel Alain¹,Wright John J.¹,Kramer Robert¹,Langley David R.¹,Vyas Dolatrai M.¹

Affiliation:

1. The Bristol-Myers Squibb Pharmaceutical Research Institute, 5 Research Parkway, Wallingford, Connecticut 06492, The Bristol-Myers Squibb Pharmaceutical Research Institute, P.O. Box 4000, Princeton, New Jersey 08543, and The Bristol-Myers Squibb Pharmaceutical Research Institute, Candiac, QC, Canada J5R 1J1

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049090z

Reference24 articles.

1. Fluorescence Polarization Studies of the Binding of BMS 181176 to DNA

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