A Remote Secondary Binding Pocket Promotes Heteromultivalent Targeting of DC-SIGN

Author:

Wawrzinek Robert1,Wamhoff Eike-Christian12ORCID,Lefebre Jonathan12,Rentzsch Mareike12,Bachem Gunnar3,Domeniconi Gary3,Schulze Jessica12,Fuchsberger Felix F.12,Zhang Hengxi12,Modenutti Carlos4,Schnirch Lennart12,Marti Marcelo A.4ORCID,Schwardt Oliver5,Bräutigam Maria1,Guberman Mónica1,Hauck Dirk67,Seeberger Peter H.12,Seitz Oliver3ORCID,Titz Alexander678ORCID,Ernst Beat5ORCID,Rademacher Christoph12910ORCID

Affiliation:

1. Department of Biomolecular Systems, Max Planck Institute of Colloids and Interfaces, 14424 Potsdam, Germany

2. Department of Chemistry and Biochemistry, Freie University of Berlin, 14195 Berlin, Germany

3. Department of Chemistry, Humboldt University of Berlin, 12489 Berlin, Germany

4. Departamento de Química Biológica e IQUIBICEN-CONICET, Universidad de Buenos Aires, C1428EHA Ciudad de Buenos Aires, Argentina

5. Department of Pharmaceutical Sciences, University of Basel, 4056 Basel, Switzerland

6. Chemical Biology of Carbohydrates, Helmholtz Institute for Pharmaceutical Research Saarland, Helmholtz Centre for Infection Research, 66123 Saarbrücken, Germany

7. German Centre for Infection Research, Campus Hannover-Braunschweig, 38124 Braunschweig, Germany

8. Department of Chemistry, Saarland University, 66123 Saarbrücken, Germany

9. University of Vienna, Department of Pharmaceutical Sciences, Althanstrasse 14, 1090 Vienna, Austria

10. University of Vienna, Department of Microbiology, Immunology and Genetics, Max F. Perutz Laboratories, Biocenter 5, 1030 Vienna, Austria

Funder

Deutscher Akademischer Austauschdienst

Deutsche Forschungsgemeinschaft

Boehringer Ingelheim Stiftung

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

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