Screening and Phenotypical Characterization of Schistosoma mansoni Histone Deacetylase 8 (SmHDAC8) Inhibitors as Multistage Antischistosomal Agents

Author:

Saccoccia Fulvio1,Brindisi Margherita2ORCID,Gimmelli Roberto1,Relitti Nicola3ORCID,Guidi Alessandra1,Saraswati A Prasanth3,Cavella Caterina3,Brogi Simone34ORCID,Chemi Giulia3ORCID,Butini Stefania3,Papoff Giuliana1,Senger Johanna5,Herp Daniel5,Jung Manfred5ORCID,Campiani Giuseppe3ORCID,Gemma Sandra3ORCID,Ruberti Giovina1ORCID

Affiliation:

1. Institute of Biochemistry and Cell Biology (IBBC), National Research Council (CNR), Campus A. Buzzati-Traverso, via E. Ramarini 32, 00015 Monterotondo (Rome), Italy

2. Department of Excellence of Pharmacy, University of Napoli Federico II, via D. Montesano 49, 80131 Naples, Italy

3. Department of Excellence of Biotechnology, Chemistry and Pharmacy, University of Siena, via Aldo Moro 2, 53100, Siena, Italy

4. Department of Pharmacy, University of Pisa, via Bonanno 6, 56126, Pisa, Italy

5. Institute of Pharmaceutical Sciences, University of Freiburg, Albertstraße 25, 79104 Freiburg, Germany

Funder

Ministero dell’Istruzione, dell’Università e della Ricerca

Deutsche Forschungsgemeinschaft

Consiglio Nazionale delle Ricerche

Collezione Nazionale di Composti Chimici e Centro di screening

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

Reference54 articles.

1. World Health Organization Schistosomiasis, 2019; available via the Internet at: https://www.who.int/schistosomiasis/en/ (accessed July 1, 2019).

2. Schistosomiasis control: praziquantel forever?

3. Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine

4. Schistosomiasis: Drugs used and treatment strategies

5. Praziquantel

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