Inhibitors of the Thioesterase Activity of Mycobacterium tuberculosis Pks13 Discovered Using DNA-Encoded Chemical Library Screening

Author:

Krieger Inna V.1,Yalamanchili Subbarao2,Dickson Paige2ORCID,Engelhart Curtis A.3,Zimmerman Matthew D4,Wood Jeremy1,Clary Ethan1,Nguyen Jasmine1,Thornton Natalie3,Centrella Paolo A.2,Chan Betty25,Cuozzo John W26ORCID,Gengenbacher Martin4,Guié Marie-Aude2,Guilinger John P2,Bienstock Corey2,Hartl Hajnalka27,Hupp Christopher D.28,Jetson Rachael29,Satoh Takashi210,Yeoman John T. S.211,Zhang Ying2,Dartois Veronique412ORCID,Schnappinger Dirk3,Keefe Anthony D.2,Sacchettini James C.1ORCID

Affiliation:

1. Department of Biochemistry & Biophysics, Texas A&M University, College Station, Texas 77843, United States

2. X-Chem Inc., 100 Beaver Street, Waltham, Massachusetts 02453, United States

3. Department of Microbiology and Immunology, Weill Cornell Medicine, New York, New York 10021, United States

4. Center for Discovery and Innovation, Hackensack Meridian Health, Nutley, New Jersey 07110, United States

5. Auron Therapeutics, 55 Chapel Street, Newton, Massachusetts 02458, United States

6. Relay Therapeutics, 399 Binney Street, Cambridge, Massachusetts 02141, United States

7. Orogen Therapeutics, 12 Gill Street, Woburn, Massachusetts 01801, United States

8. Ipsen Bioscience Inc., 1 Main Street, Cambridge, Massachusetts 02142, United States

9. Valo Health, 75 Hayden Avenue, Lexington, Massachusetts 02141, United States

10. EXO Therapeutics, 150 Cambridgepark Drive, suite 300, Cambridge, Massachusetts 02140, United States

11. Recludix Pharmaceuticals, 222 Third Street, Cambridge, Massachusetts 02142, United States

12. Hackensack Meridian School of Medicine, Hackensack Meridian Health, Nutley, New Jersey 07110, United States

Funder

Welch Foundation

Division of Intramural Research

Congressionally Directed Medical Research Programs

Bill and Melinda Gates Foundation

Publisher

American Chemical Society (ACS)

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