Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid

Author:

Bouz Ghada1ORCID,Šlechta Petr1,Jand’ourek Ondřej1,Konečná Klára1,Paterová Pavla2,Bárta Pavel1,Novák Martin13,Kučera Radim1,Dal Nils-Jørgen Knudsen4,Fenaroli Federico4ORCID,Zemanová Júlia5,Forbak Martin5,Korduláková Jana5,Pavliš Oto6,Kubíčková Pavla6,Doležal Martin1,Zitko Jan1ORCID

Affiliation:

1. Faculty of Pharmacy in Hradec Králové, Charles University, Heyrovského 1203, Hradec Králové 500 05, Czech Republic

2. Department of Clinical Microbiology, University Hospital, Sokolská 581, Hradec Králové 500 05, Czech Republic

3. Biomedical Research Center, University Hospital Hradec Kralove, Sokolská 581, Hradec Králové 500 05, Czech Republic

4. Department of Biosciences, University of Oslo, Blindernveien 31, Oslo 0371, Norway

5. Department of Biochemistry, Faculty of Natural Sciences, Comenius University in Bratislava, Mlynská Dolina, Ilkovičova 6, Bratislava 84215, Slovakia

6. Military Health Institute, Military Medical Agency, Tychonova 1, Prague 6 160 01, Czech Republic

Funder

European Regional Development Fund

Grantov? Agentura Cesk? Republiky

European Food Safety Authority

Ministerstvo Zdravotnictv? Cesk? Republiky

Univerzita Karlova v Praze

Fakultn? nemocnice Hradec Kr?lov?

Agent?ra na Podporu V?skumu a V?voja

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

Cited by 1 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献

1. Comprehensive coverage on anti-mycobacterial endeavour reported during 2022;European Journal of Medicinal Chemistry;2023-07

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