7-N-Substituted-3-oxadiazole Quinolones with Potent Antimalarial Activity Target the Cytochrome bc1 Complex

Author:

Nguyen William12,Dans Madeline G.12,Currie Iain12,Awalt Jon Kyle12ORCID,Bailey Brodie L.12,Lumb Chris1,Ngo Anna1,Favuzza Paola12,Palandri Josephine12,Ramesh Saishyam3,Penington Jocelyn12ORCID,Jarman Kate E.12,Mukherjee Partha4,Chakraborty Arnish4,Maier Alexander G.3,van Dooren Giel G.3,Papenfuss Tony12,Wittlin Sergio56ORCID,Churchyard Alisje7,Baum Jake78,Winzeler Elizabeth A.9ORCID,Baud Delphine10,Brand Stephen10,Jackson Paul F.11,Cowman Alan F.12,Sleebs Brad E.12ORCID

Affiliation:

1. The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia

2. Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia

3. Research School of Biology, The Australian National University, Canberra 2600, Australia

4. TCG Lifesciences, Kolkata, West Bengal 700091, India

5. Swiss Tropical and Public Health Institute, Kreuzstrasse 2, 4123 Allschwil, Switzerland

6. University of Basel, 4003 Basel, Switzerland

7. Department of Life Sciences, Imperial College London, South Kensington, SW7 2AZ U.K.

8. School of Biomedical Sciences, University of New South Wales, Sydney 2031, Australia

9. School of Medicine, University of California San Diego, 9500 Gilman Drive 0760, La Jolla, California 92093, United States

10. Medicines for Malaria Venture, Geneva 1215, Switzerland

11. Global Public Health, Janssen R&D LLC, La Jolla, California 92121, United States

Funder

Department of Health, State Government of Victoria

National Health and Medical Research Council

Australian Cancer Research Foundation

Wellcome

Australian Government

Medicines for Malaria Venture

University of Melbourne

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

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