Inhibitors of Acyl-CoA:Cholesterol O-Acyl Transferase (ACAT) as Hypocholesterolemic Agents. CI-1011: An Acyl Sulfamate with Unique Cholesterol-Lowering Activity in Animals Fed Noncholesterol-Supplemented Diets-Reference-Cited by-同舟云学术

Inhibitors of Acyl-CoA:Cholesterol O-Acyl Transferase (ACAT) as Hypocholesterolemic Agents. CI-1011: An Acyl Sulfamate with Unique Cholesterol-Lowering Activity in Animals Fed Noncholesterol-Supplemented Diets

Published:1996-01-01 Issue:26 Volume:39 Page:5031-5034
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lee Helen T.¹,Sliskovic Drago R.¹,Picard Joseph A.¹,Roth Bruce D.¹,Wierenga Wendell¹,Hicks James L.¹,Bousley Richard F.¹,Hamelehle Katherine L.¹,Homan Reynold¹,Speyer Cecilia¹,Stanfield Richard L.¹,Krause Brian R.¹

Affiliation:

1. Departments of Medicinal Chemistry, Radiochemistry, and Vascular and Cardiac Diseases, Parke-Davis Pharmaceutical Research, Division of Warner-Lambert Company, 2800 Plymouth Road, Ann Arbor, Michigan 48105

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960674d

Reference21 articles.

1. Inhibitors of Acyl-CoA:cholesterol O-Acyl Transferase (ACAT) as Hypocholesterolemic Agents.6.The First Water-Soluble ACAT Inhibitor with Lipid-Regulating Activity

2. Hepatic microsomal induction profile of carbamic acid [[2,6-bis(1-methylethyl)phenoxy] sulfonyl]-2,6-bis(1-methylethyl) phenyl ester, monosodium salt (PD138142-15), a novel lipid regulating agent

3. Inhibitors of Acyl-CoA:Cholesterol O-Acyltransferase. 17. Structure−Activity Relationships of Several Series of Compounds Derived from N-Chlorosulfonyl Isocyanate

4. Hedayatullah, M.; Hugeny, J.C. Synthèses A L'Aide D'Hetérocumulènes. 4. Action L'Isocyanate De Chlorosulfonyle Sur les Phénols Encombrés. (Syntheses using Heterocumulenes. 4. Reaction of N-chlorosulfonyl Isocyanate with Hindered Phenols.)Phosphorus Sulfur1984,19, 167−172.

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