Rational Targeting of Active-Site Tyrosine Residues Using Sulfonyl Fluoride Probes-Reference-Cited by-同舟云学术

Rational Targeting of Active-Site Tyrosine Residues Using Sulfonyl Fluoride Probes

Published:2015-01-29 Issue:4 Volume:10 Page:1094-1098
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Hett Erik C.¹²,Xu Hua¹²,Geoghegan Kieran F.¹²,Gopalsamy Ariamala¹²,Kyne Robert E.¹²,Menard Carol A.¹²,Narayanan Arjun¹²,Parikh Mihir D.¹²,Liu Shenping¹²,Roberts Lee¹²,Robinson Ralph P.¹²,Tones Michael A.¹²,Jones Lyn H.¹²

Affiliation:

1. Worldwide Medicinal Chemistry and ‡Rare Disease Research Unit, Pfizer, 610 Main Street, Cambridge, Massachusetts 02139, United States

2. Structural Biology and Biophysics, Worldwide Medicinal Chemistry, ∥Worldwide Medicinal Chemistry, and ⊥Primary Pharmacology Group, Pfizer, Eastern Point Road, Groton, Connecticut 06340, United States

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cb5009475

Reference35 articles.

1. Can the flow of medicines be improved? Fundamental pharmacokinetic and pharmacological principles toward improving Phase II survival

2. Target validation using chemical probes

3. In-cell click labelling of small molecules to determine subcellular localisation

4. Small Molecules Targeting Hepatitis C Virus-Encoded NS5A Cause Subcellular Redistribution of Their Target: Insights into Compound Modes of Action

Cited by 157 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The Modular Synthesis of Sulfondiimidoyl Fluorides and their Application to Sulfondiimidamide and Sulfondiimine Synthesis;Angewandte Chemie International Edition;2024-08-19

2. The Modular Synthesis of Sulfondiimidoyl Fluorides and their Application to Sulfondiimidamide and Sulfondiimine Synthesis;Angewandte Chemie;2024-08-19

3. A Convenient One-Pot Process for Converting Thiols into Sulfonyl Fluorides Using H2O2 as an Oxidant;Synthesis;2024-07-19

4. Sulfur (VI) fluoride exchange (SuFEx): a versatile tool to profile protein-biomolecule interactions for therapeutic development;Medicinal Chemistry Research;2024-06-18

5. Tying the knot with lysine;Nature Reviews Chemistry;2024-03-18