Stepwise Modulation of Neurokinin-3 and Neurokinin-2 Receptor Affinity and Selectivity in Quinoline Tachykinin Receptor Antagonists-Reference-Cited by-同舟云学术

Stepwise Modulation of Neurokinin-3 and Neurokinin-2 Receptor Affinity and Selectivity in Quinoline Tachykinin Receptor Antagonists

Published:2001-04-25 Issue:11 Volume:44 Page:1675-1689
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Blaney Frank E.¹,Raveglia Luca F.¹,Artico Marco¹,Cavagnera Stefano¹,Dartois Catherine¹,Farina Carlo¹,Grugni Mario¹,Gagliardi Stefania¹,Luttmann Mark A.¹,Martinelli Marisa¹,Nadler Guy M. M. G.¹,Parini Carlo¹,Petrillo Paola¹,Sarau Henry M.¹,Scheideler Mark A.¹,Hay Douglas W. P.¹,Giardina Giuseppe A. M.¹

Affiliation:

1. Department of Computational & Structural Sciences, SmithKline Beecham Pharmaceuticals, New Frontiers Science Park, Third Avenue, Harlow, Essex, England CM19 5AW, Departments of Medicinal Chemistry and Neurobiology Research, SmithKline Beecham S.p.A., Via Zambeletti, 20021 Baranzate, Milano, Italy, SmithKline Beecham Laboratoires Pharmaceutiques, Unité de Recherche, 4, rue du ChesnayBeauregard, Boite Postale 96205, F-35762 St. Gregoire, France, and Department of Pulmonary Biology, SmithKline Beecham...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000501v

Reference63 articles.

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