Use of a Pharmacophore Model for the Design of EGFR Tyrosine Kinase Inhibitors: Isoflavones and 3-Phenyl-4(1H)-quinolones-Reference-Cited by-同舟云学术

Use of a Pharmacophore Model for the Design of EGFR Tyrosine Kinase Inhibitors: Isoflavones and 3-Phenyl-4(1H)-quinolones

Published:1999-02-26 Issue:6 Volume:42 Page:1018-1026
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Traxler Peter¹,Green Jennifer¹,Mett Helmut¹,Séquin Urs¹,Furet Pascal¹

Affiliation:

1. NOVARTIS Pharmaceuticals, Therapeutic Area Oncology, NOVARTIS Limited, CH-4002 Basel, Switzerland, and Institute of Organic Chemistry, University of Basel, CH-4056 Basel, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm980551o

Reference35 articles.

1. Growth Factors and Cancer

2. Tyrosine Kinase Inhibition: An Approach to Drug Development

3. Signal transduction by receptors with tyrosine kinase activity

4. Overexpression of Transforming Growth Factor α in Psoriatic Epidermis

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