Design, Synthesis, and Evaluation of Su- gar Amino Acid Based Inhibitors of Pro- tein Prenyl Transferases PFT and PGGT-1-Reference-Cited by-同舟云学术

Design, Synthesis, and Evaluation of Su- gar Amino Acid Based Inhibitors of Pro- tein Prenyl Transferases PFT and PGGT-1

Published:2004-06-24 Issue:16 Volume:47 Page:3920-3923
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

El Oualid Farid¹,Burm Brigitte E. A.¹,Leroy Ingrid M.¹,Cohen Louis H.¹,van Boom Jacques H.¹,van den Elst Hans¹,Overkleeft Herman S.¹,van der Marel Gijs A.¹,Overhand Mark¹

Affiliation:

1. Leiden Institute of Chemistry, Gorlaeus Laboratories, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands, and TNO Prevention and Health, Gaubius Laboratory, P.O. Box 2215, 2301 CE Leiden, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049927q

Reference57 articles.

1. Farnesyltransferase inhibitors: antineoplastic properties, mechanisms of action, and clinical prospects

2. Perspectives on farnesyl transferase inhibitors in cancer therapy

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