Indolylarylsulfones Bearing Natural and Unnatural Amino Acids. Discovery of Potent Inhibitors of HIV-1 Non-Nucleoside Wild Type and Resistant Mutant Strains Reverse Transcriptase and Coxsackie B4 Virus-Reference-Cited by-同舟云学术

Indolylarylsulfones Bearing Natural and Unnatural Amino Acids. Discovery of Potent Inhibitors of HIV-1 Non-Nucleoside Wild Type and Resistant Mutant Strains Reverse Transcriptase and Coxsackie B4 Virus

Published:2009-03-12 Issue:7 Volume:52 Page:1922-1934
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Piscitelli Francesco¹,Coluccia Antonio¹,Brancale Andrea¹,La Regina Giuseppe¹,Sansone Anna¹,Giordano Cesare¹,Balzarini Jan¹,Maga Giovanni¹,Zanoli Samantha¹,Samuele Alberta¹,Cirilli Roberto¹,La Torre Francesco¹,Lavecchia Antonio¹,Novellino Ettore¹,Silvestri Romano¹

Affiliation:

1. Istituto Pasteur-Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, Piazzale Aldo Moro 5, I-00185 Roma, Italy, Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff, CF10 3NB, U.K., Istituto di Chimica Biomolecolare del CNR, Sapienza Università di Roma, Piazzale Aldo Moro 5, I-00185 Roma, Italy, Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, Via Domenico Montesano 49, I-80131, Napoli,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm801470b

Reference51 articles.

1. WHO/UNAIDS. 2007AIDS epidemic update.

2. HIV drug development: the next 25 years

3. Toward Improved Anti-HIV Chemotherapy: Therapeutic Strategies for Intervention with HIV Infections

4. Highlights in the Development of New Antiviral Agents

Cited by 60 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Exploration of carboxamide hybrid indolyl aryl sulfones as antiretroviral agents by HIV-1 reverse transcriptase inhibition and antioxidant effects: Synthesis, biochemical screening and computational analysis;Journal of Molecular Structure;2025-01

2. Deciphering the enigmas of non‐nucleoside reverse transcriptase inhibitors (NNRTIs): A medicinal chemistry expedition towards combating HIV drug resistance;Medicinal Research Reviews;2024-08-26

3. Exploration of Carboxamide Hybrid Indolyl Aryl Sulfones for HIV by Hiv-1 Reverse Transcriptase Inhibition and Antioxidant Effects: Synthesis, Biochemical Screening and Computational Analysis;2024

4. Visible-Light-Mediated Regioselective Chlorosulfonylation of Acrylamides;Synthesis;2023-03-23

5. Design, Synthesis and In Vitro Evaluation of Spirooxindole-Based Phenylsulfonyl Moiety as a Candidate Anti-SAR-CoV-2 and MERS-CoV-2 with the Implementation of Combination Studies;International Journal of Molecular Sciences;2022-10-06