Stereoselective Addition of 2-Phenyloxazol-4-yl Trifluoromethanesulfonate to N-Sulfinyl Imines: Application to the Synthesis of the HCV Protease Inhibitor Boceprevir-Reference-Cited by-同舟云学术

Stereoselective Addition of 2-Phenyloxazol-4-yl Trifluoromethanesulfonate to N-Sulfinyl Imines: Application to the Synthesis of the HCV Protease Inhibitor Boceprevir

Published:2012-12-20 Issue:2 Volume:78 Page:706-710
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Morris William J.¹,Muppalla Kiran K.¹,Cowden Cameron¹,Ball Richard G.¹

Affiliation:

1. Department of Process Research, Merck Research Laboratories, Rahway, New Jersey 07065, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo301856f

Reference51 articles.

1. New Pharmacotherapy for Hepatitis C

2. Protease inhibitors for the treatment of chronic hepatitis C genotype-1 infection: the new standard of care

3. Diagnosis, management, and treatment of hepatitis C: An update

4. Control of Hepatitis C: A Medicinal Chemistry Perspective

5. Challenges in Modern Drug Discovery: A Case Study of Boceprevir, an HCV Protease Inhibitor for the Treatment of Hepatitis C Virus Infection

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