Synthesis and Evaluation of Estrogen Agonism of Diaryl 4,5-Dihydroisoxazoles, 3-Hydroxyketones, 3-Methoxyketones, and 1,3-Diketones: A Compound Set Forming a 4D Molecular Library-Reference-Cited by-同舟云学术

Synthesis and Evaluation of Estrogen Agonism of Diaryl 4,5-Dihydroisoxazoles, 3-Hydroxyketones, 3-Methoxyketones, and 1,3-Diketones: A Compound Set Forming a 4D Molecular Library

Published:2008-06-01 Issue:12 Volume:51 Page:3562-3571
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Pulkkinen Juha T.¹,Honkakoski Paavo¹,Peräkylä Mikael¹,Berczi Istvan¹,Laatikainen Reino¹

Affiliation:

1. Laboratories of Chemistry, Biochemistry, Department of Biosciences, University of Kuopio, P.O. Box 1627, FIN-70211 Kuopio, Finland, Department of Pharmaceutics, University of Kuopio, P.O. Box 1627, FIN-70211 Kuopio, Finland, Department of Immunology, Faculty of Medicine, University of Manitoba, Winnipeg, Manitoba R3E 0W3, Canada

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm8001795

Reference72 articles.

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3. Novel Ligands that Function as Selective Estrogens or Antiestrogens for Estrogen Receptor-α or Estrogen Receptor-β*

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