Development of a New Practical Synthesis of a 5-HT2C Receptor Agonist-Reference-Cited by-同舟云学术

Development of a New Practical Synthesis of a 5-HT2C Receptor Agonist

Published:2010-11-02 Issue:6 Volume:14 Page:1438-1447
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Gontcharov Alexander¹,Shaw Chia-Cheng¹,Yu Qing¹,Tadayon Sam¹,Bernatchez Michel¹,Lankau Mark¹,Cantin Michel¹,Potoski John¹,Khafizova Gulnaz¹,Stack Gary¹,Gross Jonathan¹,Zhou Dahui¹

Affiliation:

1. Wyeth Research Chemical Development and Chemical Sciences, 401 North Middletown Road, Pearl River, New York 10965, United States, Wyeth Research, Chemical Development, 1025 Marcel Laurin Boulevard, St. Laurent, QC H4R 1J6, Canada, and Wyeth Research, Chemical Sciences, 865 Ridge Road, Monmouth Junction, New Jersey 08852, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op100233f

Reference29 articles.

1. 5-HT2C receptor agonists as an innovative approach for psychiatric disorders

2. U.S. Patent 7,435,837, 2008

3. The process in Scheme1has been successfully scaled up to 70 g for preparation of1and its des-fluoro analogue (unpublished results).

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