Mechanism and Site of Inhibition of AMPA Receptors: Pairing a Thiadiazole with a 2,3-Benzodiazepine Scaffold
Author:
Affiliation:
1. Department of Chemistry, and Center for Neuroscience Research, University at Albany, SUNY, Albany, New York 12222, United States
2. CF Pharma Pharmaceutical Manufacturing Co., Ltd, H-1097 Budapest, Kén utca 5, Hungary
Publisher
American Chemical Society (ACS)
Subject
Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/cn400193u
Reference58 articles.
1. Electrophysiological studies with a 2,3-benzodiazepine muscle relaxant: GYKI 52466
2. Non-competitive AMPA Antagonists of 2,3-Benzodiazepine Type
3. New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists
4. synthesis and Structure-Activity Relationships of 2,3-Benzodiazepines as AMPA Receptor Antagonists
5. Quinoxalinediones: Potent Competitive Non-NMDA Glutamate Receptor Antagonists
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