Structure−Activity Relationship of Quinoline Derivatives as Potent and Selective α2C-Adrenoceptor Antagonists-Reference-Cited by-同舟云学术

Structure−Activity Relationship of Quinoline Derivatives as Potent and Selective α2C-Adrenoceptor Antagonists

Published:2006-09-28 Issue:21 Volume:49 Page:6351-6363
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Höglund Iisa P. J.¹,Silver Satu¹,Engström Mia T.¹,Salo Harri¹,Tauber Andrei¹,Kyyrönen Hanna-Kaisa¹,Saarenketo Pauli¹,Hoffrén Anna-Marja¹,Kokko Kurt¹,Pohjanoksa Katariina¹,Sallinen Jukka¹,Savola Juha-Matti¹,Wurster Siegfried¹,Kallatsa Oili A.¹

Affiliation:

1. Juvantia Pharma Ltd, Lemminkäisenkatu 5, FI-20520 Turku, Finland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060262x

Reference35 articles.

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2. Gene targeting — homing in on α2-adrenoceptor-subtype function

3. Distribution of α2-adrenergic receptor subtype gene expression in rat brain

4. Distribution of ?2C-adrenergic receptor-like immunoreactivity in the rat central nervous system

5. Evaluation of the α2C-adrenoceptor as a neuropsychiatric drug target

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