Modulation of Activity Profiles for Largazole-Based HDAC Inhibitors through Alteration of Prodrug Properties-Reference-Cited by-同舟云学术

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Modulation of Activity Profiles for Largazole-Based HDAC Inhibitors through Alteration of Prodrug Properties

Published:2014-07-07 Issue:8 Volume:5 Page:905-910
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Salvador Lilibeth A.¹,Park Heekwang²,Al-Awadhi Fatma H.,Liu Yanxia,Kim Bumki²,Zeller Sabrina L.²,Chen Qi-Yin,Hong Jiyong²³,Luesch Hendrik

Affiliation:

1. Marine Science Institute, College of Science, University of the Philippines, Diliman, Quezon City 1101, Philippines

2. Department of Chemistry, Duke University, Durham, North Carolina 27708, United States

3. Department of Pharmacology and Cancer Biology, Duke University Medical Center, Durham, North Carolina 27710, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml500170r

Reference24 articles.

1. Epigenetics in cancer

2. Increased expression of histone deacetylase 2 is found in human gastric cancer

3. HDAC Inhibitors and Other Histone Modifying Natural Products as Emerging Anticancer Agents

4. Dimethyl sulfoxide to vorinostat: development of this histone deacetylase inhibitor as an anticancer drug

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