Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone: A Potent, Orally Bioavailable Human CB1/CB2 Dual Agonist with Antihyperalgesic Properties and Restricted Central Nervous System Penetration-Reference-Cited by-同舟云学术

Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone: A Potent, Orally Bioavailable Human CB1/CB2 Dual Agonist with Antihyperalgesic Properties and Restricted Central Nervous System Penetration

Published:2007-07-14 Issue:16 Volume:50 Page:3851-3856
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Dziadulewicz Edward K.¹,Bevan Stuart J.¹,Brain Christopher T.¹,Coote Paul R.¹,Culshaw Andrew J.¹,Davis Andrew J.¹,Edwards Lee J.¹,Fisher Adrian J.¹,Fox Alyson J.¹,Gentry Clive¹,Groarke Alex¹,Hart Terance W.¹,Huber Werner¹,James Iain F.¹,Kesingland Adam¹,La Vecchia Luigi¹,Loong Yvonne¹,Lyothier Isabelle¹,McNair Kara¹,O'Farrell Cathal¹,Peacock Marcus¹,Portmann Robert¹,Schopfer Ulrich¹,Yaqoob Mohammed¹,Zadrobilek Jiri¹

Affiliation:

1. Novartis Institutes for BioMedical Research, 5 Gower Place, London WC1E 6BS, United Kingdom, and Novartis Pharma AG, CH-4002, Basel, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm070317a

Reference43 articles.

1. Dancing with Antipodes: (Bipolar Illness-in Memory of My Mother)

2. Marijuana and Medicine: Assessing the Science Base: A Summary of the 1999 Institute of Medicine Report

3. The endocannabinoid nervous system

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