General Solid-Phase Synthesis Approach To Prepare Mechanism-Based Aspartyl Protease Inhibitor Libraries. Identification of Potent Cathepsin D Inhibitors-Reference-Cited by-同舟云学术

General Solid-Phase Synthesis Approach To Prepare Mechanism-Based Aspartyl Protease Inhibitor Libraries. Identification of Potent Cathepsin D Inhibitors

Published:1998-09-01 Issue:38 Volume:120 Page:9735-9747
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Lee Christina E.¹,Kick Ellen K.¹,Ellman Jonathan A.¹

Affiliation:

1. Contribution from the Department of Chemistry, University of California, Berkeley, California 94720

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja981812m

Reference44 articles.

1. Molecular Recognition of Protein−Ligand Complexes: Applications to Drug Design

2. Structure and Function of the Aspartic Proteinases

3. Aspartic Proteinases

4. Discovery of protease inhibitors using targeted libraries

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