Structure Guided Design of 5-Arylindazole Glucocorticoid Receptor Agonists and Antagonists-Reference-Cited by-同舟云学术

Structure Guided Design of 5-Arylindazole Glucocorticoid Receptor Agonists and Antagonists

Published:2010-05-14 Issue:11 Volume:53 Page:4531-4544
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Yates Christopher M.¹,Brown Peter J.¹,Stewart Eugene L.¹,Patten Christopher²,Austin Robert J. H.²,Holt Jason A.¹,Maglich Jodi M.¹,Angell Davina C.²,Sasse Rosemary Z.¹,Taylor Simon J.²,Uings Iain J.²,Trump Ryan P.¹

Affiliation:

1. Molecular Discovery Research, GlaxoSmithKline, Research Triangle Park, North Carolina 27709-3398

2. Drug Discovery, GlaxoSmithKline, Gunnels Wood Road, Stevenage, SG1 2NY, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100447c

Reference47 articles.

1. Mechanisms involved in the side effects of glucocorticoids

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3. Therapeutic potential of selective modulators of nuclear receptor action

4. Anti-inflammatory Actions of Glucocorticoids: Molecular Mechanisms

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